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Προβολή τεκμηρίου 
  •   Ιδρυματικό Αποθετήριο Πανεπιστημίου Θεσσαλίας
  • Επιστημονικές Δημοσιεύσεις Μελών ΠΘ (ΕΔΠΘ)
  • Δημοσιεύσεις σε περιοδικά, συνέδρια, κεφάλαια βιβλίων κλπ.
  • Προβολή τεκμηρίου
  •   Ιδρυματικό Αποθετήριο Πανεπιστημίου Θεσσαλίας
  • Επιστημονικές Δημοσιεύσεις Μελών ΠΘ (ΕΔΠΘ)
  • Δημοσιεύσεις σε περιοδικά, συνέδρια, κεφάλαια βιβλίων κλπ.
  • Προβολή τεκμηρίου
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Ιδρυματικό Αποθετήριο Πανεπιστημίου Θεσσαλίας
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  • Κοινότητες & Συλλογές
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Development of a new series of aryl ureido derivatives as anticancer agents against breast cancer cells

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Συγγραφέας
Pappas, I. S.
Ημερομηνία
2010
Λέξη-κλειδί
Aryl ureido derivatives
Breast cancer
Cancer therapy
Cell growth inhibitors
amine
bexarotene
gefitinib
isoxazole
lapatinib
paclitaxel
purine
pyrazine
pyridazine
pyridine
pyrimidine
sorafenib
thiazole
urea derivative
animal cell
antineoplastic activity
breast carcinoma
cancer cell culture
cancer chemotherapy
CMT U27 cell
conference paper
controlled study
drug synthesis
nonhuman
Εμφάνιση Μεταδεδομένων
Επιτομή
Breast cancer is the second cause of cancer mortality worldwide in humans and half of all tumours in dogs and there is an unmet need for novel anticancer agents. I have developed a new series of aryl ureido derivatives as anticancer agents. These compounds have a strong antiproliferative effect against canine breast cancer CMT-U27 cells at concentrations (1-10 μM) comparable to drugs that have already been used in chemotherapy such as gefitinib, soferanib and lapatinib. These results suggest that aryl ureido derivatives were potent inhibitors of proliferation of breast cancer cells. © PHARMAKON-Press.
URI
http://hdl.handle.net/11615/32016
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  • Δημοσιεύσεις σε περιοδικά, συνέδρια, κεφάλαια βιβλίων κλπ. [19674]

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