dc.creator | Kalavrizioti, D. | en |
dc.creator | Vourekas, A. | en |
dc.creator | Tekos, A. | en |
dc.creator | Tsagla, A. | en |
dc.creator | Stathopoulos, C. | en |
dc.creator | Drainas, D. | en |
dc.date.accessioned | 2015-11-23T10:31:00Z | |
dc.date.available | 2015-11-23T10:31:00Z | |
dc.date.issued | 2003 | |
dc.identifier | 10.1023/A:1022290110116 | |
dc.identifier.issn | 3014851 | |
dc.identifier.uri | http://hdl.handle.net/11615/28757 | |
dc.description.abstract | A cell-free system derived from Dictyostelium discoideum has been used to study the kinetics of inhibition of RNase P by puromycin, amicetin and blasticidin S. Detailed kinetic analysis showed that the type of inhibition of RNase P activity by puromycin is simple competitive, whereas the type of inhibition by amicetin and blasticidin S is simple non-competitive. On the basis of Ki values amicetin is stronger inhibitor than puromycin and blasticidin S. | en |
dc.source | Molecular Biology Reports | en |
dc.source.uri | http://www.scopus.com/inward/record.url?eid=2-s2.0-0037335175&partnerID=40&md5=2df686e55f0be5c3b51e0e1f6dd27821 | |
dc.subject | Protein synthesis inhibitors | en |
dc.subject | Ribozymes | en |
dc.subject | RNase P | en |
dc.subject | amicetin | en |
dc.subject | antibiotic agent | en |
dc.subject | blasticidin S | en |
dc.subject | peptidyltransferase | en |
dc.subject | puromycin | en |
dc.subject | ribonuclease P | en |
dc.subject | unclassified drug | en |
dc.subject | article | en |
dc.subject | cell free system | en |
dc.subject | competitive inhibition | en |
dc.subject | concentration response | en |
dc.subject | controlled study | en |
dc.subject | enzyme activity | en |
dc.subject | enzyme inhibition | en |
dc.subject | kinetics | en |
dc.subject | nonhuman | en |
dc.subject | Animals | en |
dc.subject | Dictyostelium | en |
dc.subject | Dose-Response Relationship, Drug | en |
dc.subject | Endoribonucleases | en |
dc.subject | Nucleosides | en |
dc.subject | Peptidyl Transferases | en |
dc.subject | Pyrimidine Nucleosides | en |
dc.subject | RNA, Catalytic | en |
dc.subject | Dictyostelium discoideum | en |
dc.subject | Protozoa | en |
dc.title | Kinetics of inhibition of ribonuclease P activity by peptidyltransferase inhibitors: Effect of antibiotics on RNase P | en |
dc.type | journalArticle | en |